发明名称 |
6-SUBSTITUTED HEXAHYDROINDAZOLO (7,6,5,-1J) ISOQUINOLINES AND HEXAHYDROISOINDOLO (4,5,6,-1J) ISOQUINOLINES |
摘要 |
<p>6-Substituted hexahydroindazolo or hexahydroisoindolo isoquinolines, having dopamine agonist and dopamine antagonist activity, are described herein. The compounds are prepared by reacting the corresponding 8-dimethylaminomethylene derivative with a substituted amine. Novel intermediates are also disclosed.</p> |
申请公布号 |
CA1182457(A) |
申请公布日期 |
1985.02.12 |
申请号 |
CA19820398593 |
申请日期 |
1982.03.17 |
申请人 |
LILLY (ELI) AND COMPANY |
发明人 |
KORNFELD, EDMUND C.;BACH, NICHOLAS J.;TITUS, ROBERT D. |
分类号 |
C07D471/04;A61K31/47;A61K31/473;A61K31/4745;A61P9/12;A61P25/00;A61P25/08;A61P25/16;C07D217/14;C07D217/16;C07D221/14;C07D471/06;(IPC1-7):C07D471/04 |
主分类号 |
C07D471/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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