发明名称 |
PHENYLETHANOLAMINOTETRALINCARBOXAMID-DERIVATE |
摘要 |
The present invention relates to a phenylethanolaminotetralincarboxamide derivative represented by the general formula: <CHEM> (wherein A represents a lower alkylene group; B represents an amino group, a di(lower alkyl)amino group or a 3 to 7-membered alicyclic amino group which may contain an oxygen atom in the ring; the carbon atom marked with * represents a carbon atom in (R) configuration, (S) configuration or a mixture thereof; and the carbon atom marked with (S) represents a carbon atom in (S) configuration) and a pharmaceutically acceptable salt thereof, which have a selective beta 2-adrenergic receptor stimulating effect with relieved burdens on the heart such as tachycardia and are useful as an agent for the prevention of threatened abortion and premature labor, a bronchodilator, and an agent for pain remission and promoting stone removal in urolithiasis. |
申请公布号 |
DE69736924(D1) |
申请公布日期 |
2006.12.21 |
申请号 |
DE1997636924 |
申请日期 |
1997.04.04 |
申请人 |
KISSEI PHARMACEUTICAL CO. LTD. |
发明人 |
KITAZAWA, MAKIO;OKAZAKI, KOSUKE;TAMAI, TETSURO;SAITO, MASARU;TANAKA, NOBUYUKI;KOBAYASHI, HIROAKI;KIKUCHI, KEN;MURANAKA, HIDEYUKI |
分类号 |
C07C235/06;A61K31/165;A61K31/445;A61K31/495;A61K31/535;C07D295/16;C07D295/18;C07D295/185 |
主分类号 |
C07C235/06 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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