发明名称 PHENYLETHANOLAMINOTETRALINCARBOXAMID-DERIVATE
摘要 The present invention relates to a phenylethanolaminotetralincarboxamide derivative represented by the general formula: <CHEM> (wherein A represents a lower alkylene group; B represents an amino group, a di(lower alkyl)amino group or a 3 to 7-membered alicyclic amino group which may contain an oxygen atom in the ring; the carbon atom marked with * represents a carbon atom in (R) configuration, (S) configuration or a mixture thereof; and the carbon atom marked with (S) represents a carbon atom in (S) configuration) and a pharmaceutically acceptable salt thereof, which have a selective beta 2-adrenergic receptor stimulating effect with relieved burdens on the heart such as tachycardia and are useful as an agent for the prevention of threatened abortion and premature labor, a bronchodilator, and an agent for pain remission and promoting stone removal in urolithiasis.
申请公布号 DE69736924(D1) 申请公布日期 2006.12.21
申请号 DE1997636924 申请日期 1997.04.04
申请人 KISSEI PHARMACEUTICAL CO. LTD. 发明人 KITAZAWA, MAKIO;OKAZAKI, KOSUKE;TAMAI, TETSURO;SAITO, MASARU;TANAKA, NOBUYUKI;KOBAYASHI, HIROAKI;KIKUCHI, KEN;MURANAKA, HIDEYUKI
分类号 C07C235/06;A61K31/165;A61K31/445;A61K31/495;A61K31/535;C07D295/16;C07D295/18;C07D295/185 主分类号 C07C235/06
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