发明名称 TRIAZOLOPYRIDINES
摘要 The present invention relates to triazolopyridine compounds of general formula (I) which are Monopolar Spindle 1 kinase (Mps-1 or TTK) inhibitors: Formula (I), in which R1, R2, R3, R4, and R5 are as given in the description and in the claims, to methods of preparing said compounds, to pharmaceutical compositions and combinations comprising said compounds, to the use of said compounds for manufacturing a pharmaceutical composition for the treatment or prophylaxis proliferative of diseases, as well as to intermediate compounds useful in the preparation of said compounds.
申请公布号 US2012328610(A1) 申请公布日期 2012.12.27
申请号 US201013512701 申请日期 2010.11.17
申请人 SCHULZE VOLKER;KOPPITZ MARCUS;KOSEMUND DIRK;SCHIROK HARTMUT;BADER BENJAMIN;LIENAU PHILIP;WENGNER ANTJE MARGRET;BRIEM HANS;HOLTON SIMON;SIEMEISTER GERHARD;PRECHTL STEFAN;BOEMER ULF;BAYER INTELLECTUAL PROPERTY GMBH 发明人 SCHULZE VOLKER;KOPPITZ MARCUS;KOSEMUND DIRK;SCHIROK HARTMUT;BADER BENJAMIN;LIENAU PHILIP;WENGNER ANTJE MARGRET;BRIEM HANS;HOLTON SIMON;SIEMEISTER GERHARD;PRECHTL STEFAN;BOEMER ULF
分类号 A61K31/437;A61K31/444;A61K31/4545;A61K31/4745;A61K31/496;A61K31/513;A61K31/519;A61K31/52;A61K31/5377;A61K31/567;A61K31/573;A61K31/664;A61K31/69;A61K31/704;A61K31/7068;A61K31/7076;A61K33/24;A61K38/14;A61K39/395;A61P35/00;A61P35/02;A61P35/04;C07D471/04 主分类号 A61K31/437
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