发明名称 |
TETRAHYDROTHIAZOLOPYRIDINE INHIBITORS OF PHOSPHATIDYLINOSITOL 3-KINASE |
摘要 |
The present invention relates to compounds useful as inhibitors of PI3K, particularly of PI3Kγ. The invention also provides pharmaceutically acceptable compositions comprising said compounds and methods of using the compositions in the treatment of various disease, conditions, or disorders. |
申请公布号 |
US2012039849(A1) |
申请公布日期 |
2012.02.16 |
申请号 |
US201113211502 |
申请日期 |
2011.08.17 |
申请人 |
ARONOV ALEX;BANDARAGE UPUL KEERTHI;COTTRELL KEVIN MICHAEL;DAVIES ROBERT J.;KRUEGER ELAINE B.;LEDEBOER MARK WILLEM;LEDFORD BRIAN;LE TIRAN ARNAUD;MESSERSMITH DAVID;WANG TIANSHENG;XU JINWANG;LIAO YUSHENG;VERTEX PHARMACEUTICALS INCORPORATED |
发明人 |
ARONOV ALEX;BANDARAGE UPUL KEERTHI;COTTRELL KEVIN MICHAEL;DAVIES ROBERT J.;KRUEGER ELAINE B.;LEDEBOER MARK WILLEM;LEDFORD BRIAN;LE TIRAN ARNAUD;MESSERSMITH DAVID;WANG TIANSHENG;XU JINWANG;LIAO YUSHENG |
分类号 |
A61K31/437;A61K31/497;A61K38/07;A61K38/21;A61K39/395;A61P25/00;A61P29/00;A61P37/02;A61P37/06;C07D471/04;C12N9/99 |
主分类号 |
A61K31/437 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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