SUBSTITUTED ARYLSULFONYLAMINOMETHYLPHOSPHONIC ACID DERIVATIVES, THEIR PREPARATION AND THEIR USE IN THE TREATMENT OF TYPE I AND II DIABETES MELLITUS,申请号US20080669979-传众专利搜索

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发明名称	SUBSTITUTED ARYLSULFONYLAMINOMETHYLPHOSPHONIC ACID DERIVATIVES, THEIR PREPARATION AND THEIR USE IN THE TREATMENT OF TYPE I AND II DIABETES MELLITUS
摘要	The present invention relates to substituted arylsulphonylaminomethyl-phosphonic acid derivatives of general formula wherein R, X, Y and Z are defined as in claim 1, the tautomers, enantiomers, diastereomers, mixtures thereof and salts thereof which have valuable pharmacological properties, particularly the suppression of the interaction of glycogen phosphorylase a with the GL subunit of glycogen-associated protein phosphatase 1 (PP1), and their use as pharmaceutical compositions.
申请公布号	US2010210595(A1)	申请公布日期	2010.08.19
申请号	US20080669979	申请日期	2008.07.25
申请人	BOEHRINGER INGELHEIM INTERNATIONAL GMBH	发明人	WAGNER HOLGER;LANGKOPF ELKE;ECKHARDT MATTHIAS;STREICHER RUEDIGER;SCHOELCH CORINNA;SCHULER-METZ ANNETTE;PAUTSCH ALEXANDER
分类号	A61K31/675;A61K31/683;A61P3/10;C07F9/572;C07F9/59;C07F9/6509;C07F9/653;C07F9/6533;C07F9/6541;C07F9/6558	主分类号	A61K31/675
代理机构		代理人
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