发明名称 |
3, 4-DIHYDROQUINOLIN-2 ( 1H ) -ONE DERIVATIVES AS SODIUM CHANNEL MODULATORS |
摘要 |
The present invention relates to sodium channel inhibitors of Formula (I): in which R1, R2, R3, R4, R5, R6, and R7 are as defined above, and to their use in the treatment of various disease states, including cardiovascular diseases and diabetes. |
申请公布号 |
WO2010074807(A1) |
申请公布日期 |
2010.07.01 |
申请号 |
WO2009US62386 |
申请日期 |
2009.10.28 |
申请人 |
GILEAD PALO ALTO, INC.;ABELMAN, MATTHEW;CHU, NANCY;JIANG, ROBERT;LEUNG, KWAN;ZABLOCKI, JEFF |
发明人 |
ABELMAN, MATTHEW;CHU, NANCY;JIANG, ROBERT;LEUNG, KWAN;ZABLOCKI, JEFF |
分类号 |
C07D413/06;A61K31/4704;A61K31/4709;A61P3/10;A61P9/00;C07D215/227;C07D417/06 |
主分类号 |
C07D413/06 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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