发明名称 3, 4-DIHYDROQUINOLIN-2 ( 1H ) -ONE DERIVATIVES AS SODIUM CHANNEL MODULATORS
摘要 The present invention relates to sodium channel inhibitors of Formula (I): in which R1, R2, R3, R4, R5, R6, and R7 are as defined above, and to their use in the treatment of various disease states, including cardiovascular diseases and diabetes.
申请公布号 WO2010074807(A1) 申请公布日期 2010.07.01
申请号 WO2009US62386 申请日期 2009.10.28
申请人 GILEAD PALO ALTO, INC.;ABELMAN, MATTHEW;CHU, NANCY;JIANG, ROBERT;LEUNG, KWAN;ZABLOCKI, JEFF 发明人 ABELMAN, MATTHEW;CHU, NANCY;JIANG, ROBERT;LEUNG, KWAN;ZABLOCKI, JEFF
分类号 C07D413/06;A61K31/4704;A61K31/4709;A61P3/10;A61P9/00;C07D215/227;C07D417/06 主分类号 C07D413/06
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