发明名称 Method for Producing 4(3H)-Quinazolinone Derivative
摘要 This invention is related to a method for producing 3-{4-[3-(1-pyrrolidinyl)propoxy]phenyl}-5-trifluoromethyl-4(3H)-quinazolinone comprising a step for reacting 2-methyl-5-trifluoromethyl-4H-3,1-benzoxazin-4-one with 4-[3-(1-pyrrolidinyl)propoxy]aniline or an acid-addition salt thereof, or 4-(1-cyclobutyl-4-piperidinoy9oxyaniline or acid addition salt thereof in the presence of an acid catalyst.
申请公布号 US2009131664(A1) 申请公布日期 2009.05.21
申请号 US20060922479 申请日期 2006.07.04
申请人 AKAO ATSUSHI;IIDA TAKEHIKO;ITOH TAKAHIRO;MASE TOSHIAKI;SATO KIMIHIKO;SAWADA NAOTAKA;KADOWAKI CHIE;TSURITANI TAKAYUKI;YASUDA NOBUYOSHI 发明人 AKAO ATSUSHI;IIDA TAKEHIKO;ITOH TAKAHIRO;MASE TOSHIAKI;SATO KIMIHIKO;SAWADA NAOTAKA;KADOWAKI CHIE;TSURITANI TAKAYUKI;YASUDA NOBUYOSHI
分类号 C07D401/02 主分类号 C07D401/02
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