发明名称 |
METHOD FOR SYNTHESIS OF (S)-AZIRIDINE-2-CARBOXYAMIDE AND (R)-AZIRIDINE-2-CARBOXYAMIDE, AND INTERMEDIATE PRODUCTS OF SYNTHESIS |
摘要 |
There is worked out a novel method for synthesis (S)-aziridine-2-carboxyamide and (R)-aziridine-2-carboxyamide, that provides obtaining both enantiomers by one scheme from (R)- or (S)-methyl-1-tritylaziridine-2-carboxylate by one-top technology process with high-percentage yield of products having outstanding superiority of enantiomers. There are offered new intermediate products for obtaining chiral-type of aziridine-2-carboxyamide. |
申请公布号 |
LV13848(A) |
申请公布日期 |
2009.01.20 |
申请号 |
LV20080000188 |
申请日期 |
2008.11.03 |
申请人 |
PHARMIDEA, SIA |
发明人 |
TURKS M&Amacr,RIS;ZIC&Amacr,NE DAINA;RIJKURE INESE |
分类号 |
C07D203/00;A61K31/396 |
主分类号 |
C07D203/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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