| 发明名称 |
Novel methods for the preparation of taxanes using oxazolidine intermediates |
| 摘要 |
Novel oxazolidines finding utility as intermediates in the preparation of C-13 acyloxy sidechain-bearing taxanes such as paclitaxel and analogs thereof. The present invention also relates to novel methods of coupling the oxazolidines to form the aforementioned taxanes, and to methods of preparing the oxazolidines.
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| 申请公布号 |
US2002161238(A1) |
申请公布日期 |
2002.10.31 |
| 申请号 |
US20010014950 |
申请日期 |
2001.12.11 |
| 申请人 |
THOTTATHIL JOHN K.;TRIFUNOVICH IVAN D. |
发明人 |
THOTTATHIL JOHN K.;TRIFUNOVICH IVAN D. |
| 分类号 |
C07C227/12;C07C229/22;C07C231/12;C07C233/82;C07C233/87;C07D263/04;C07D263/06;C07D305/14;C07D413/12;C07F7/18;(IPC1-7):C0735/14;C0747/02 |
主分类号 |
C07C227/12 |
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