发明名称 BENZOTHIAZINE DIOXIDE DERIVATIVES
摘要 Compounds of the formula: <CHEM> wherein R1 is 2-pyridyl, 6-methyl-2-pyridyl, 6-fluoro-2-pyridyl, 6-chloro-2-pyridyl, 5-methyl-3-isoxazolyl, 2-thiazolyl, 5-methyl-2-thiazolyl, 1-oxo-2,4,6-cycloheptatrien-2-yl phenyl, nitrophenyl or mono- or disubstituted phenyl wherein each substituent is fluorine, chlorine, bromine, trifluoromethyl, alkyl having from one to three carbon atoms or alkoxy having from one to three carbon atoms; R2 is hydrogen, alkanoyl having from two to six carbon atoms, benzoyl, p-chlorobenzoyl, toluoyl, thenoyl, furoyl, -COR3 or COOR3 wherein R3 is alkyl having from one to eight carbon atoms; and n is an integer of from three to five. These compounds are useful as analgesics or antiinflammatory agents.
申请公布号 PH22947(A) 申请公布日期 1989.02.03
申请号 PH19570000352 申请日期 1987.05.14
申请人 PFIZER INC. 发明人 LOMBARDINO JOSEPH GEORGE;MARFAT ANTHONY
分类号 A61K31/54;A61P29/00;C07D279/02;C07D417/12;C07D417/14 主分类号 A61K31/54
代理机构 代理人
主权项
地址