发明名称 |
SNTHRACYCLINE DISACCHARIDES |
摘要 |
<p>Anthracycline disaccharides having antitumor activity are prepared by condensing N-trifluoroacetyldaunomycin with a 1-halosugar in the presence of a silver salt such as AgSO3CF3 as catalyst to form a protected di-glycoside which upon mild alkaline hydrolysis yields the novel disaccharides.</p> |
申请公布号 |
GB1561507(A) |
申请公布日期 |
1980.02.20 |
申请号 |
GB19760047835 |
申请日期 |
1976.11.17 |
申请人 |
SOC FARMACEUTICI ITALIA SPA |
发明人 |
PENCO SERGIO;FRANCHI GIULIANO;ARCAMONE FEDERICO |
分类号 |
A61K31/65;A61P35/00;C07H15/252;(IPC1-7):07H15/24;61K31/70 |
主分类号 |
A61K31/65 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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