发明名称 |
Thiazinoindoles useful as antidepressants |
摘要 |
Thiazinoindole derivatives characterized by having an amino(lower)alkyl radical attached to the 1 position of a 1H-1,4-thiazino[4,3-a]indole nucleus are disclosed. The amino portion of the amino(lower)alkyl radical may be further substituted with one or two lower alkyl groups or incorporated in a heterocyclic amine radical. The derivatives are substituted further at positions 1 and 10 and may be optionally substituted at positions 3, 4, 6, 7, 8 and 9. The thiazinoindole derivatives of this invention are useful antidepressant and antiulcer agents. Methods for the use of these derivatives and compositions containing them are also disclosed.
|
申请公布号 |
US4066763(A) |
申请公布日期 |
1978.01.03 |
申请号 |
US19760750293 |
申请日期 |
1976.12.13 |
申请人 |
AYERST MCKENNA AND HARRISON LTD. |
发明人 |
DEMERSON, CHRISTOPHER A.;HUMBER, LESLIE G.;SANTROCH, GEORGE;DOBSON, THOMAS A.;JIRKOVSKY, IVO |
分类号 |
C07D209/08;(IPC1-7):C07D513/04;A61K31/38 |
主分类号 |
C07D209/08 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|