发明名称 |
Penicillins and processes for their preparation and use |
摘要 |
6-[ alpha -(Imidazolidin-2-on-1-carbonylamido)acetamido]-penicillanic acids substituted in the 3-position of the imidazolidinone ring with phenyl or a substituted phenyl group and on the alpha -carbon atom of the acetamido bridge with a phenyl, thienyl, cyclohexenyl or cyclohexadienyl group, and their salts, are antibacterial agents. The compounds, of which alpha -(3-phenylimidazolidin-2-on-1-ylcarbonylamino)benzylpenicillin is a representative example, are prepared by acylation of the corresponding 6-( alpha -aminoacetamido)penicillanic acid or a derivative thereof.
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申请公布号 |
US4031229(A) |
申请公布日期 |
1977.06.21 |
申请号 |
US19760692930 |
申请日期 |
1976.06.04 |
申请人 |
BAYER AKTIENGESELLSCHAFT |
发明人 |
KONIG, HANS-BODO;METZGER, KARL GEORG;SCHROCK, WILFRIED |
分类号 |
C07D499/10;C07D233/32;C07D233/38;C07D499/00;C07D499/04;C07D499/64;C07D499/66;C07D499/68;C07D499/70;(IPC1-7):A61K31/43 |
主分类号 |
C07D499/10 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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