发明名称 |
7,8,9,10-tetrahydro-6H-azepino, 6,7,8,9-tetrahydro-pyrido and 2,3-dihydro-2H-pyrrolo[2,1-b]-quinazolinone derivatives |
摘要 |
Disclosed herein are 7,8,9,10-tetrahydro-6H-azepino, 6,7,8,9-tetrahydro-pyrido and 2,3-dihydro-2H-pyrrolo[2,1-b]-quinazolinone derivatives of formula (I) and their use as active ingredients in the preparation of pharmaceutical compositions, wherein the variables are as defined in the specification. Also disclosed are processes for the preparation of the compounds of formula (I), pharmaceutical compositions containing one or more of those compounds and especially their use as orexin receptor antagonists.
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申请公布号 |
NZ538029(A) |
申请公布日期 |
2006.08.31 |
申请号 |
NZ20030538029 |
申请日期 |
2003.07.08 |
申请人 |
ACTELION PHARMACEUTICALS LTD |
发明人 |
AISSAOUI, HAMED;CLOZEL, MARTINE;FISCHLI, WALTER;KOBERSTEIN, RALF;SIFFERLEN, THIERRY;WELLER, THOMAS |
分类号 |
A61K31/519;A61K31/522;A61K45/00;A61P3/04;A61P9/00;A61P25/18;A61P25/20;A61P25/24;A61P35/00;A61P43/00;C07D471/04;C07D487/04;(IPC1-7):A61K31/519 |
主分类号 |
A61K31/519 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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