发明名称 BICYCLIC OXAZINE AND THIAZINE OXAZOLIDINONE ANTIBACTERIALS
摘要 PCT No. PCT/US95/12751 Sec. 371 Date May 14, 1997 Sec. 102(e) Date May 14, 1997 PCT Filed Oct. 31, 1995 PCT Pub. No. WO96/15130 PCT Pub. Date May 23, 1996Phenyloxazolidinone compound of formula (I)or a pharmaceutically acceptable salt thereof characterized by a bicyclic thiazine or oxazine substituent. The compounds are useful antimicrobial agents, effective against a number of human and veterinary pathogens, including gram-positive aerobic bacteria such as multiply-resistant staphylococci, streptococci and enterococci as well as anaerobic organisms such as Bacteroides spp. and Clostridia spp. species, and acid-fast organisms such as Mycobacterium tuberculosis, Mycobacterium avium and Mycobacterium spp.
申请公布号 NZ295528(A) 申请公布日期 1999.03.29
申请号 NZ19950295528 申请日期 1995.10.31
申请人 PHARMACIA & UPJOHN CO 发明人 BARBACHYN, MICHAEL R;THOMAS, RICHARD C;CLEEK, GARY J;THOMASCO, LISA MARIE;GADWOOD, ROBERT C
分类号 A61K31/535;A61K31/537;A61K31/54;A61P31/00;A61P31/04;C07D491/04;C07D491/048;C07D491/08;C07D495/04;C07D495/08;(IPC1-7):C07D513/20;C07D498/18;A61K31/42 主分类号 A61K31/535
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