发明名称 FUSED PYRAZOLE DERIVATIVE HAVING AUTOTAXIN INHIBITORY ACTIVITY
摘要 The present invention provides a compound that has an autotaxin inhibitory effect and is represented by formula (I) (in the formula, R1, R2, R3, R4a, R4b, R5a, and R5b are as defined in the description.), a medicine that uses said compound as an active component, and a treatment or prevention method for a disease involving autotaxin, said treatment or prevention method being characterized by the administration of said compound.
申请公布号 WO2015129821(A1) 申请公布日期 2015.09.03
申请号 WO2015JP55693 申请日期 2015.02.26
申请人 THE UNIVERSITY OF TOKYO;TOHOKU UNIVERSITY;SHIONOGI & CO., LTD. 发明人 NAGANO, TETSUO;OKABE, TAKAYOSHI;KOJIMA, HIROTATSU;KAWAGUCHI, MITSUYASU;NUREKI, OSAMU;ISHITANI, RYUICHIRO;NISHIMASU, HIROSHI;AOKI, JUNKEN;FUJIKOSHI, CHIAKI;KATOU, MANABU;ODAN, MASAHIDE;TANAKA, NOBUYUKI;TATENO, YUSUKE;YAMANE, JUNJI
分类号 C07D487/04;A61K31/4985;A61K31/5377;A61K31/55;A61P1/16;A61P9/00;A61P9/10;A61P11/00;A61P13/02;A61P13/12;A61P17/00;A61P17/02;A61P19/02;A61P21/00;A61P25/00;A61P25/04;A61P27/02;A61P29/00;A61P35/00;A61P37/06;C07D487/18;C07D491/048 主分类号 C07D487/04
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