发明名称 |
NOVEL ESTERS OF 4, 9-DIHYDROXY-NAPHTHO [2, 3-b] FURANS FOR DISEASE THERAPIES |
摘要 |
The present invention discloses esters of 4,9-dihydroxy-naphtho[2,3-b]furans and methods of making and using the same. The present invention also discloses conversion of the esters into therapeutically active 4,9-dihydroxy-naphtho[2,3-b]furans in vivo. The present invention furthermore discloses pharmaceutical compositions comprising the esters of 4,9-dihydroxy-naphtho[2,3-b]furans for the treatment of various indications including proliferative diseases. |
申请公布号 |
US2013345176(A1) |
申请公布日期 |
2013.12.26 |
申请号 |
US201114002986 |
申请日期 |
2011.03.04 |
申请人 |
JIANG ZHIWEI;WANG AIJIN;HU HONGWEI;XU JIALI;HU YUESONG;LI XIAN;YE YAN;WANG JIE;LI QINGLONG;ZHOUSHAN HAIZHONGZHOU XINSHENG PHARMACEUTICALS CO., LTD. |
发明人 |
JIANG ZHIWEI;WANG AIJIN;HU HONGWEI;XU JIALI;HU YUESONG;LI XIAN;YE YAN;WANG JIE;LI QINGLONG |
分类号 |
C07D307/92;A61K31/343;A61K31/665;A61K45/06;C07F9/655 |
主分类号 |
C07D307/92 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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