发明名称 6-Substituted 2,3,4,5-Tetrahydro-1H-Benzo [d]Azepines as 5-HT2C Receptor Agonists
摘要 <p>The present invention provides 6-substituted 2,3,4,5-tetrahydro-1H-benzo[d]azepines of Formula I as selective 5-HT 2C receptor agonists for the treatment of 5-HT 2C associated disorders including obesity, obsessive/compulsive disorder, depression, and anxiety: where: R 6 is -S-L-R 15 and other substituents are as defined in the specification.</p>
申请公布号 EP2479168(A1) 申请公布日期 2012.07.25
申请号 EP20120161584 申请日期 2005.02.18
申请人 ELI LILLY AND COMPANY 发明人 ALLEN, JOHN, GORDON;TIDWELL, MICHAEL, WADE;VICTOR, FRANTZ;WILLIAMS, ANDREW CAERWYN;ZHANG, DEYI;BOYD, STEVEN, ARMEN;CONWAY, RICHARD, GERARD;DEO, ARUNDHATI, S;LEE, WAI-MAN;SIEDEM, CHRISTOPHER, STEPHEN;SINGH, AJAY;BRINER, KARIN;COHEN, MICHAEL, PHILIP;GALKA, CHRISTOPHER, STANLEY;HELLMAN, SARAH, LYNNE;MARTINEZ-GRAU, MARIA ANGELES;REINHARD, MATTHEW, ROBERT;RODRIGUEZ, MICHAEL, JOHN;ROTHHAAR, ROGER, RYAN
分类号 C07D223/16;A61K31/55;A61P3/04;A61P25/22;A61P25/24;A61P25/30;C07D401/12;C07D403/06;C07D403/12;C07D405/12;C07D409/12;C07D413/12;C07D413/14;C07D417/06;C07D417/12 主分类号 C07D223/16
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