发明名称 |
SALTS OF ISOBUTYRIC ACID (1 R*, 2R*, 4R* ) -2- (2-{ [3- (4, 7-DIMETH0XY-1 H-BENZOIMIDAZOL-2-YL) -PROPYL] -METHYL-AMINO } -ETHYL) -5-PHENYL-BICYCLO [2.2.2] OCT-5- EN- 2 -YL. |
摘要 |
<p>The invention relates to crystalline salts of isobutyric acid (1R*,2R*,4R*)-2-(2-{[3-(4,7-dimethoxy-1H-benzoimidazol-2-yl)-pr opyl]-methyl-amino}-ethyl)-5-phenyl-bicyclo[2.2.2]oct-5-en-2-yl ester, processes for the preparation thereof, pharmaceutical compositions containing said crystalline salts, and their use as medicaments, especially as calcium channel blockers.</p> |
申请公布号 |
MX2011004138(A) |
申请公布日期 |
2011.07.20 |
申请号 |
MX20110004138 |
申请日期 |
2009.10.21 |
申请人 |
ACTELION PHARMACEUTICALS LTD. |
发明人 |
KURT HILPERT;FRANCIS HUBLER;STEFAN ABELE;DORTE RENNEBERG;MARKUS VON RAUMER;STEPHANIE COMBES;JACQUES-ALEXIS FUNEL;KATHARINA REICHENBAECHER |
分类号 |
C07D235/14;A61K31/4184;A61P9/00 |
主分类号 |
C07D235/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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