发明名称 APPLICATION OF THIENOPYRIDONE DERIVATIVES AS AMPA-ACTIVATORS AND PHARMACEUTIC COMPOSITIONS, CONTAINING THEM
摘要 FIELD: medicine, pharmaceutics. ^ SUBSTANCE: invention relates to application of thienopyridone derivatives of formula (I), in which B represents CH, represents , or , R represents H, R1 and R2, independently on each other, represent H, linear or branched (C1-C4)alkyl, (C1-C4)cycloalkyl, halogen or together form group -(CH2)n-, where n=1- 4, R3 and R4, independently on each other, represent H, R6 represents H, X represents -O-, or their pharmaceutically acceptable salts for preparation of pharmaceutical composition. ^ EFFECT: obtaining pharmaceutical composition, suitable for treatment of diabetes, metabolic syndrome and obesity. ^ 8 cl, 1 tbl, 210 ex
申请公布号 RU2416409(C2) 申请公布日期 2011.04.20
申请号 RU20080109914 申请日期 2006.07.03
申请人 MERK PATENT GMBKH 发明人 ALLAKUBOZE SOFI;SHARON KRISTIN;KHOKK B'ERN;PESHKE OLIVER
分类号 A61K31/4436;A61P3/10;C07D495/04 主分类号 A61K31/4436
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