发明名称 PROCESS FOR SUBSTITUTED 3-AMINO-5-OXO-4,5-DIHYDRO-[1,2,4]TRIAZINES
摘要 Processes including preparation of trans-4-[(3-amino-5-oxo-4,5-dihydro-[1,2,4]triazin-6-ylmethyl)-carbamoyl]-cyclohexanecarboxylic acid methyl ester, and its conversion to trans-4-(4-amino-5-susbtituted-imidazo[5,1- ][1,2,4]triazin-7-yl)-cyclohexanecarboxylic acid compounds.
申请公布号 WO2011005909(A2) 申请公布日期 2011.01.13
申请号 WO2010US41278 申请日期 2010.07.08
申请人 OSI PHARMACEUTICALS, INC.;DONG, HANQING;MAO, YUNYU;MULVIHILL, KRISTEN, MICHELLE;RECHKA, JOSEF, A.;WERNER, DOUGLAS, S. 发明人 DONG, HANQING;MAO, YUNYU;MULVIHILL, KRISTEN, MICHELLE;RECHKA, JOSEF, A.;WERNER, DOUGLAS, S.
分类号 C07D253/06;C07D403/04;C07D487/04 主分类号 C07D253/06
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