发明名称 Substituted pyrazolopyrimidines, methods for the production thereof, use of the same for controlling pathogenic fungi, and agents containing said compounds
摘要 The invention relates to substituted pyrazolopyrimidines of formula (I) wherein the substituents have the following designations: L represents halogen, alkyl, halogenalkyl, alkenyl, alkoxy, amino, NHR, NR<SUB>2</SUB>, cyano, S(-O)<SUB>n</SUB>A<SUP>1 </SUP>or C(-O)A<SUP>2</SUP>, R representing alkyl or alkylcarbonyl, A<SUP>1 </SUP>representing hydrogen, hydroxy, alkyl, alkylamino or dialkylamino, n representing 0, 1 or 2, and A<SUP>2 </SUP>representing alkenyl, alkoxy, halogenalkoxy or one of the groups cited for A<SUP>1</SUP>; m represents 0 or 1 to 5; R<SUP>1 </SUP>represents alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, alkadienyl, halogenalkenyl, cycloalkenyl, alkinyl, halogenalkinyl or cycloalkinyl, phenyl, naphthyl, or a five-membered to ten-membered saturated, partially unsaturated or aromatic heterocycle containing between one and four heteroatoms from the group O, N or S; and R<SUP>2 </SUP>represents hydrogen or one of the groups cited for R<SUP>1</SUP>. Together with the nitrogen atom to which they are bonded, R<SUP>1 </SUP>and R<SUP>2 </SUP>can form a five-membered to six-membered ring that can be interrupted by an atom from the groups O, N and S, and R<SUP>1 </SUP>and/or R<SUP>2 </SUP>can also be substituted according to the description. Furthermore, in formula (I): X represents halogen, cyano, OH, alkyl, alkoxy or halogenalkoxy; Y represents a five-membered to ten-membered saturated, partially unsaturated or aromatic heterocycle according to the description, or a group X or another group according to the description; p represents 1 or 2, the groups Y being potentially different when p=2; and p represents 0, when X is according to the description. The invention also relates to methods and intermediate products for producing said compounds, agents containing the same, and the use thereof for controlling phytopathogenic fungi.
申请公布号 US2006258685(A1) 申请公布日期 2006.11.16
申请号 US20050558251 申请日期 2005.11.21
申请人 WAGNER OLIVIER;GROTE THOMAS;BLETTNER CARSTEN;GEWEHR MARKUS;GRAMMENOS WASSILIOS;GYPSER ANDREAS;MULLER BERND;RHEINHEIMER JOACHIM;SCHAFER PETER;SCHIEWECK FRANK;SCHWOGLER ANJA;BLASCO JORDI T I;AKERS ALAN;SPEAKMAN JOHN-BRYAN;RACK MICHAEL;STIERL REINHARD;SCHERER MARIA;SCHOFL ULRICH;STRATHMANN SIEGFRIED 发明人 WAGNER OLIVIER;GROTE THOMAS;BLETTNER CARSTEN;GEWEHR MARKUS;GRAMMENOS WASSILIOS;GYPSER ANDREAS;MULLER BERND;RHEINHEIMER JOACHIM;SCHAFER PETER;SCHIEWECK FRANK;SCHWOGLER ANJA;BLASCO JORDI T.I.;AKERS ALAN;SPEAKMAN JOHN-BRYAN;RACK MICHAEL;STIERL REINHARD;SCHERER MARIA;SCHOFL ULRICH;STRATHMANN SIEGFRIED
分类号 A61K31/519;A01N43/90;C07D487/04 主分类号 A61K31/519
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