发明名称 |
NOVEL CYCLOSPORINS |
摘要 |
Cyclosporins wherein the residue at the 1-position has the formula I <IMG> in which -x-y- is -CH=CH-(trans) or -CH2-CH2-, X is 0 or S and R is hydrogen, optionally halo or hydroxy substituted- C1-3-alkyl, -alkoxy or -alkylthio, or amino or mono- or di- (C1-2alkyl)-amino, useful as pharmaceuticals, in particular for asthma therapy.
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申请公布号 |
CA2090634(C) |
申请公布日期 |
2005.12.13 |
申请号 |
CA19932090634 |
申请日期 |
1993.03.01 |
申请人 |
BOELSTERLI, JOHANN JAKOB;EBERLE, MARCEL KARL;NAEF, RETO;PAYNE, TREVOR GLYN |
发明人 |
BOELSTERLI, JOHANN JAKOB;EBERLE, MARCEL KARL;NAEF, RETO;PAYNE, TREVOR GLYN |
分类号 |
A61K38/00;A61K38/13;A61P11/00;A61P29/00;A61P37/06;C07K1/113;C07K7/64;(IPC1-7):C07K7/64 |
主分类号 |
A61K38/00 |
代理机构 |
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代理人 |
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地址 |
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