发明名称 |
Serine protease inhibitors |
摘要 |
Compounds of formula (I) in which R2, X, Y, Cy, L and Lp(D)n have the meanings given in the specification, are inhibitors of the serine protease, Factor Xa and are useful in the treatment of cardiovascular disorders. |
申请公布号 |
US2004242656(A1) |
申请公布日期 |
2004.12.02 |
申请号 |
US20040876672 |
申请日期 |
2004.06.28 |
申请人 |
LIEBESCHUETZ JOHN WALTER;MURRAY CHRISTOPHER WILLIAM;YOUNG STEPHEN CLINTON;CAMP NICHOLAS PAUL;JONES STUART DONALD;WYLIE WILLIAM ALEXANDER;MASTERS JOHN JOSEPH;WILEY MICHAEL ROBERT;SHEEHAN SCOTT MARTIN;ENGEL DAVID BIRENBAUM;WATSON BRIAN MORGAN |
发明人 |
LIEBESCHUETZ JOHN WALTER;MURRAY CHRISTOPHER WILLIAM;YOUNG STEPHEN CLINTON;CAMP NICHOLAS PAUL;JONES STUART DONALD;WYLIE WILLIAM ALEXANDER;MASTERS JOHN JOSEPH;WILEY MICHAEL ROBERT;SHEEHAN SCOTT MARTIN;ENGEL DAVID BIRENBAUM;WATSON BRIAN MORGAN |
分类号 |
A61K31/40;A61K31/4439;A61K31/445;A61K31/4545;A61K31/4709;A61P1/16;A61P7/02;A61P9/02;A61P9/10;A61P11/00;A61P11/06;A61P17/00;A61P17/02;A61P19/02;A61P29/00;A61P35/00;A61P43/00;C07D207/12;C07D211/46;C07D401/12;C07D401/14;C07D417/14;(IPC1-7):A61K31/44;A61K31/19;A61K31/165 |
主分类号 |
A61K31/40 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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