发明名称 |
SELECTIVE LINEAR PEPTIDES WITH MELANOCORTIN-4 RECEPTOR (MC4-R) AGONIST ACTIVITY |
摘要 |
The present invention relates to peptides comprising the structure (S1) wherein R<1>, R<6>, R<7>, R<8>, m, n, A and B are as defined in the description and claims. Such compounds selectively activate melanocortin-4 (MC-4) receptor activity.
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申请公布号 |
WO0174844(A3) |
申请公布日期 |
2002.06.13 |
申请号 |
WO2001EP03529 |
申请日期 |
2001.03.27 |
申请人 |
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发明人 |
CHEN, LI;CHEUNG, ADRIAN, WAI-HING;CHU, XIN-JIE;DANHO, WALEED;SWISTOK, JOSEPH;YAGALOFF, KEITH, ALAN |
分类号 |
A61K38/00;A61K38/08;A61P3/04;A61P5/00;A61P43/00;C07K1/04;C07K5/107;C07K5/117;C07K7/02;C07K7/06;C07K14/68;(IPC1-7):C07K14/68;A61K38/07;A61K38/34 |
主分类号 |
A61K38/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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