发明名称 CRISTALLINE ( - ) - 3R,4R -TRANS-7-METHOXY -2,2-DIMETHYL-3-PHENYL-4- {4-[2-(PYRROLIDIN-1-YL)ETHOXY] PHENYL}CHROMANE, HYDROGEN MALEATE
摘要 The present invention provides novel crystalline ( - ) - 3R,4R -trans-7-methoxy -2,2-dimethyl-3-phenyl-4- {4-[2-(pyrrolidin-1-yl)ethoxyl] phenyl}chromane, hydrogen maleate useful for reducing or preventin bone loss as well as pharmaceutical compositions containing the same. A process for preparing ( - ) - 3R,4R -trans-7-methoxy-2,2-dimethyl-3-phenyl-4-{4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}chromane, hydrogen maleate is described.
申请公布号 WO9856782(A1) 申请公布日期 1998.12.17
申请号 WO1998DK00244 申请日期 1998.06.11
申请人 NOVO NORDISK A/S 发明人 TREPPENDAHL, SVEND;JENSEN, KLAUS, SNEJ;MCGRAW, SCOTT, EUGENE
分类号 C07D311/58;(IPC1-7):C07D311/58;A61K31/40;A61K31/35 主分类号 C07D311/58
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