发明名称 |
HETEROCYCLIC DERIVATIVES OF AMINES OR THEIR PHARMACEUTICALLY ACCEPTABLE SALTS, INTERMEDIATE COMPOUNDS, PHARMACEUTICAL COMPOSITION, METHOD OF INHIBITION OF CHOLINE ESTERASE ACTIVITY, METHOD OF SYNTHESIS OF COMPOUNDS |
摘要 |
<p>FIELD: chemistry of heterocyclic compounds. SUBSTANCE: invention relates to heterocyclic derivatives of amines of the formula (I) <EMI ID=0.107 HE=21 WI=57 TI=CHI> where X, Y, M, L and R<SP>1</SP>,R<SP>2</SP>,R<SP>7</SP>,R are given in description, or their salts and intermediate compounds. Invention relates to also pharmaceutical composition and a method of inhibition of choline esterase activity based on compounds of the formula (I) and a method of synthesis of these compounds. EFFECT: improved method of synthesis. 10 cl, 1 tbl, 38 ex</p> |
申请公布号 |
RU2119920(C1) |
申请公布日期 |
1998.10.10 |
申请号 |
RU19930055137 |
申请日期 |
1992.03.09 |
申请人 |
EHJSAJ KO., LTD. |
发明人 |
ANABELLA VILLALOBOS;ARTUR ADAM NEHJDZHEL;JUPAJNG LIANG CHEN |
分类号 |
A61K31/415;A61K31/41;A61K31/425;A61K31/4427;A61K31/445;A61K31/451;A61K31/4523;A61K31/47;A61K31/472;A61K31/495;A61K31/496;A61K31/50;A61K31/505;A61K31/517;A61K31/53;A61K31/535;A61P25/02;A61P25/28;A61P43/00;C07D;C07D211/08;C07D211/18;C07D211/24;C07D211/30;C07D211/32;C07D211/36;C07D211/38;C07D211/60;C07D217/14;C07D231/56;C07D239/74;C07D241/42;C07D253/04;C07D261/20;C07D401/06;C07D401/12;C07D401/14;C07D409/12;C07D409/14;C07D413/06;C07D413/10;C07D413/12;C07D413/14;C07D417/06;C07D417/10;C07D417/12;C07D417/14;C07D491/056;C07D498/02;C07D498/04;C07D513/02;C07D513/04;C12N9/99;(IPC1-7):C07D413/06 |
主分类号 |
A61K31/415 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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