| 发明名称 |
GLUCOCORTICOID MIMETICS, METHODS OF MAKING THEM, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF |
| 摘要 |
Compounds of Formula (IA) wherein R1, R2, R3, R4 and R5 are as defined herein for Formula (IA), or a tautomer, prodrug, solvate, or salt thereof; pharmaceutical compositions containing such compounds, and methods of modulating the glucocorticoid receptor function and methods of treating disease-states or conditions mediated by the glucocorticoid receptor function or characterized by inflammatory, allergic, or proliferative processes in a patient using these compounds. |
| 申请公布号 |
HRP20040887(A2) |
申请公布日期 |
2005.04.30 |
| 申请号 |
HR2004P000887 |
申请日期 |
2004.09.24 |
| 申请人 |
BOEHRINGER INGELHEIM PHARMACEUTICALS INC. |
发明人 |
HIDENORI TAKAHASHI;YOUNES BEKKALI;RAJASHEKHAR BETAGERI;MARIO G. CARDOZO;THOMAS A. GILMORE;CHRISTIAN HANKE JUSTUS JOACHIM HARCKEN;THOMAS M. KIRRANE;DANIEL KUZMICH;JOHN R. PROUDFOOT;HOSSEIN RAZAVI;DORIS RIETHER;DAVID S. THOMSON;JI WANG;RENEE ZINDELL |
| 分类号 |
A61K31/343;A61K31/404;A61K31/405;A61K31/4184;A61K31/423;A61K31/437;A61K31/44;A61K31/4402;A61K31/4439;A61P1/00;A61P1/16;A61P3/04;A61P3/10;A61P5/00;A61P9/00;A61P9/10;A61P9/12;A61P17/00;A61P19/02;A61P25/00;A61P25/04;A61P27/02;A61P27/06;A61P27/16;A61P29/00;A61P35/00;A61P37/06;A61P37/08;C07C49/255;C07C49/577;C07D209/12;C07D209/30;C07D213/30;C07D213/61;C07D215/14;C07D217/16;C07D231/12;C07D233/54;C07D235/12;C07D237/08;C07D239/26;C07D241/12;C07D261/18;C07D263/32;C07D263/56;C07D277/24;C07D277/64;C07D307/80;C07D333/16;C07D401/06;C07D405/06;C07D471/04 |
主分类号 |
A61K31/343 |
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