发明名称 TRPV3 Modulators
摘要 Disclosed herein are modulators of TRPV3 of formula (I) wherein X1, X2, R1, R2, Rx, and n are as defined in the specification. Compositions comprising such compounds and methods for treating conditions and disorders using such compounds and compositions are also presented.
申请公布号 US2012245124(A1) 申请公布日期 2012.09.27
申请号 US201213428259 申请日期 2012.03.23
申请人 CLAPHAM BRUCE;COX PHIL B.;DART MICHAEL J.;GOMTSYAN ARTHUR;JINKERSON TAMMIE K.;KEDDY RYAN G.;KORT MICHAEL E.;KYM PHILIP R.;MATULENKO MARK;SCHMIDT ROBERT G.;VILLAMIL CLARA I.;VOIGHT ERIC A.;WOLLER KEVIN R.;ABBOTT LABORATORIES 发明人 CLAPHAM BRUCE;COX PHIL B.;DART MICHAEL J.;GOMTSYAN ARTHUR;JINKERSON TAMMIE K.;KEDDY RYAN G.;KORT MICHAEL E.;KYM PHILIP R.;MATULENKO MARK;SCHMIDT ROBERT G.;VILLAMIL CLARA I.;VOIGHT ERIC A.;WOLLER KEVIN R.
分类号 A61K31/4418;A61K31/444;A61K31/4545;A61K31/496;A61K31/505;A61K31/506;A61K31/5377;A61K31/541;A61K31/695;A61P29/00;C07D213/36;C07D239/26;C07D401/04;C07D401/14;C07D413/10;C07D413/12;C07D413/14;C07D417/10;C07F7/10 主分类号 A61K31/4418
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