发明名称 |
TRPV3 Modulators |
摘要 |
Disclosed herein are modulators of TRPV3 of formula (I) wherein X1, X2, R1, R2, Rx, and n are as defined in the specification. Compositions comprising such compounds and methods for treating conditions and disorders using such compounds and compositions are also presented.
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申请公布号 |
US2012245124(A1) |
申请公布日期 |
2012.09.27 |
申请号 |
US201213428259 |
申请日期 |
2012.03.23 |
申请人 |
CLAPHAM BRUCE;COX PHIL B.;DART MICHAEL J.;GOMTSYAN ARTHUR;JINKERSON TAMMIE K.;KEDDY RYAN G.;KORT MICHAEL E.;KYM PHILIP R.;MATULENKO MARK;SCHMIDT ROBERT G.;VILLAMIL CLARA I.;VOIGHT ERIC A.;WOLLER KEVIN R.;ABBOTT LABORATORIES |
发明人 |
CLAPHAM BRUCE;COX PHIL B.;DART MICHAEL J.;GOMTSYAN ARTHUR;JINKERSON TAMMIE K.;KEDDY RYAN G.;KORT MICHAEL E.;KYM PHILIP R.;MATULENKO MARK;SCHMIDT ROBERT G.;VILLAMIL CLARA I.;VOIGHT ERIC A.;WOLLER KEVIN R. |
分类号 |
A61K31/4418;A61K31/444;A61K31/4545;A61K31/496;A61K31/505;A61K31/506;A61K31/5377;A61K31/541;A61K31/695;A61P29/00;C07D213/36;C07D239/26;C07D401/04;C07D401/14;C07D413/10;C07D413/12;C07D413/14;C07D417/10;C07F7/10 |
主分类号 |
A61K31/4418 |
代理机构 |
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代理人 |
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地址 |
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