发明名称 Novel arylamidine derivative or salt thereof
摘要 An arylamidine derivative represented by a general formula described below or a salt thereof has an excellent antifungal action and high safety, and it is useful as an antifungal agent with good pharmacokinetics and pharmacodynamic properties wherein X represents an unsubstituted or substituted lower alkylene or alkenylene group; G<SUP>1 </SUP>represents an oxygen atom, a sulfur atom, or an imino group; G<SUP>2 </SUP>represents a carbon atom or a nitrogen atom; R<SUP>a </SUP>represents at least one group selected from the group consisting of a hydrogen atom, a halogen atom, and unsubstituted or substituted alkyl, cycloalkyl and alkoxy groups; R<SUP>1 </SUP>represents an unprotected or protected or unsubstituted or substituted amidino group; and R<SUP>2 </SUP>represents a substituted amino or substituted cyclic amino group, or the like.
申请公布号 US2005113424(A1) 申请公布日期 2005.05.26
申请号 US20040506422 申请日期 2004.09.02
申请人 TOYAMA CHEMICAL CO., LTD 发明人 HAYASHI KAZYUA;OJIMA KATSUJI;HORI KOZO;OKUJO NORIYUKI;MITSUYAMA JUNICHI;KUNITANI KAZUTO;TOHDO KEISUKE
分类号 A61K31/138;A61K31/44;A61P31/10;C07C257/18;C07C259/18;C07C271/64;C07C323/62;C07D207/14;C07D211/22;C07D211/26;C07D211/58;C07D213/62;C07D213/78;C07D213/85;C07D241/04;C07D241/08;C07D243/08;C07D245/02;C07D261/12;C07D295/092;C07D295/13;C07D401/06;C07D413/06;(IPC1-7):C07D213/62 主分类号 A61K31/138
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