发明名称 |
METHOD FOR PRODUCING PYRIDAZINONE DERIVATIVE AND ITS INTERMEDIATE |
摘要 |
PROBLEM TO BE SOLVED: To provide an industrially advantageous method for producing an N-(aminoalkyl)morpholine useful as an intermediate for medicines with a short step. SOLUTION: The N-(aminoalkyl)morpholine (IV) is produced in one step by reacting a compound expressed by general formula (II) with a compound expressed by general formula (III) (A<SB>1</SB>and A<SB>2</SB>are each independently a halogen; and n is an integer of 2-8). The compound (IV) is an intermediate for a pyridazinone derivative useful as medicines. COPYRIGHT: (C)2005,JPO&NCIPI
|
申请公布号 |
JP2005008604(A) |
申请公布日期 |
2005.01.13 |
申请号 |
JP20030177514 |
申请日期 |
2003.06.23 |
申请人 |
ONO PHARMACEUT CO LTD |
发明人 |
HASEGAWA TOMOYUKI;KAWANAKA YASUSHI;TAKEUCHI ATSUSHI |
分类号 |
C07D295/12;C07D237/32;(IPC1-7):C07D237/32 |
主分类号 |
C07D295/12 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|