发明名称 |
4-hydroxy-benzopyran-2-ones and 4-hydroxy-cycloalkylÝb¨pyran-2-ones useful to treat retroviral infections |
摘要 |
PCT No. PCT/US94/00938 Sec. 371 Date Aug. 4, 1995 Sec. 102(e) Date Aug. 4, 1995 PCT Filed Feb. 3, 1994 PCT Pub. No. WO94/18188 PCT Pub. Date Aug. 18, 1994The present invention relates to compounds of formula I which are 4-hydroxy-benzopyran-2-ones and 4-hydroxy-cycloalkyl[b]pyran-2-ones useful for inhibiting a retrovirus in a mammalian cell infected with said retrovirus. <IMAGE> I Wherein R10 and R20 taken together are: <IMAGE> II <IMAGE> III |
申请公布号 |
AU6166194(A) |
申请公布日期 |
1994.08.29 |
申请号 |
AU19940061661 |
申请日期 |
1994.02.03 |
申请人 |
THE UPJOHN COMPANY |
发明人 |
DAVID JOHN ANDERSON;LEE S BANITT;PAUL KOSTA TOMICH;MICHAEL JOHN BOHANON;STEVEN RONALD TURNER;JOSEPH WALTER STROHBACH;SUVIT THAISRIVONGS;CHIH-PING YANG;RICHARD CHARLES THOMAS;KAREN RENE ROMINES;PAUL ADRIAN ARISTOFF;HARVEY IRVING SKULNICK;PAUL D JOHNSON;RONALD B. GAMMILL;QINGWEI ZHANG;GORDON L. BUNDY |
分类号 |
C07D311/46;A61K31/352;A61K31/365;A61K31/37;A61K31/38;A61K31/381;A61K31/40;A61K31/4035;A61K31/404;A61K31/415;A61K31/4178;A61K31/4184;A61K31/427;A61K31/4433;A61K31/453;A61K31/4709;A61K31/496;A61K31/5377;A61P31/12;A61P31/18;A61P43/00;C07D311/54;C07D311/56;C07D311/74;C07D311/92;C07D311/94;C07D405/04;C07D405/12;C07D407/06;C07D407/08;C07D409/06;C07D409/08;C07D409/12;C07D413/12;C07D417/10;C07D417/12 |
主分类号 |
C07D311/46 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|