发明名称 2,3-DIAMINO-2,3-DIDESOXYHEXOSE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE
摘要 PCT No. PCT/EP85/00171 Sec. 371 Date Dec. 18, 1985 Sec. 102(e) Date Dec. 18, 1985 PCT Filed Apr. 17, 1985 PCT Pub. No. WO85/04881 PCT Pub. Date Nov. 7, 1985.Compounds of formula I <IMAGE> I wherein R2 and R3 are the same or different and each represent unsubstituted or substituted acyl, and (a) R1 represents lower alkyl, aralkyl or the phosphate, pyrophosphate, phosphorylethanolamine or pyrophosphorylethanolamine group, R4 represents the phosphate, pyrophosphate, phosphorylethanolamine or pyrophosphorylethanolamine group and one of R1 and R4 may additionally represent hydrogen and R5 represents hydrogen or a glycosyl radical or (b) R1 represents hydrogen, lower alkyl or aralkyl and R4 and R5 represent hydrogen, which compounds are indicated for use as pharmaceuticals, in particular as immunostimulants.
申请公布号 EP0180608(B1) 申请公布日期 1990.07.25
申请号 EP19850902023 申请日期 1985.04.17
申请人 SANDOZ AG;SANDOZ-ERFINDUNGEN VERWALTUNGSGESELLSCHAFT M.B.H.;SANDOZ-PATENT-GMBH 发明人 MACHER, INGOLF;UNGER, FRANK, MICHAEL
分类号 A61K31/70;C07D207/34;C07D207/40;C07D207/416;C07H;C07H5/06;C07H11/00;C07H11/04;C07H13/04;C07H13/06;C07H15/04;C07H15/18 主分类号 A61K31/70
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