发明名称 SALT AND MEDICAL USE
摘要 The present invention is directed to 4-[2-(5-amino-1H-pyrazol-4-yl)-4-chlorophenoxy]-5-chloro-2-fluoro-N-(1,3-thiazol-4-yl)benzenesulfonamide or a pharmaceutically acceptable salt thereof for the treatment of a disease associated with elevated blood uric acid levels, such as hyperuricemia or gout. The invention is also directed to the tosylate salt of 4-[2-(5-amino-1H-pyrazol-4-yl)-4-chlorophenoxy]-5-chloro-2-fluoro-N-(1,3-thiazol-4-yl)benzenesulfonamide.
申请公布号 HK1196535(A1) 申请公布日期 2016.10.28
申请号 HK20140109958 申请日期 2014.10.07
申请人 PFIZER LIMITED 发明人 ALI,ZAHID Z;BUTCHER,KENNETH JOHN KJ;BUTT,RICHARD PHILIP RP;FELSTEAD,STEPHER JOHN SJ;GLATT,SOPHIE S;MCKERNAN,RUTH MITCHELL RM;PANESAR,MANINDER M
分类号 A61K;A61P;C07D 主分类号 A61K
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