| 发明名称 |
TAXANE COMPOUNDS, COMPOSITIONS AND METHODS |
| 摘要 |
The present invention provides a method for the preparation of orally available pentacyclic taxane compounds, as well as intermediates useful in their preparation. |
| 申请公布号 |
US2014249186(A1) |
申请公布日期 |
2014.09.04 |
| 申请号 |
US201414199574 |
申请日期 |
2014.03.06 |
| 申请人 |
GFV, LLC |
发明人 |
THOTTATHIL JOHN K.;WARRELL RAYMOND P. |
| 分类号 |
C07D493/06 |
主分类号 |
C07D493/06 |
| 代理机构 |
|
代理人 |
|
| 主权项 |
1. A compound having the formula:
(TT)m.(HX)n.(H2O)y.(Sol)z wherein TT is tesetaxel; HX is a monobasic, dibasic, tribasic or polybasic acid; Sol is an organic solvent; m and n are each independently an integer from about 1 to about 5; and y and z are each independently an integer from 0 to about 5. |
| 地址 |
San Diego CA US |
