发明名称 FUSED IMIDAZOLE DERIVATIVE HAVING TTK INHIBITORY ACTION
摘要 Provided are a compound represented by general formula (1) and having a TTK inhibitory action and a medicine containing the compound. In formula (1), (X, Y, V, W) is (—N═, ═CR1—, ═N—, —CR7═), (—CR2═, ═N—, ═N—, —CR7═), etc.; A is an (un)substituted aromatic hydrocarbon ring, etc.; L is a single bond, —C(═O)—NRA—, etc.; Z is a group represented by the formula —NR3R4 or a group represented by the formula —OR5; R1 to R3, R6, and R7 each is a hydrogen atom, etc.; R4 and R5 each is an (un)substituted alkyl, etc.; and R8 is an (un)substituted cycloalkyl, etc.
申请公布号 US2012059162(A1) 申请公布日期 2012.03.08
申请号 US201113192369 申请日期 2011.07.27
申请人 KUSAKABE KEN-ICHI;YOSHIDA HIROSHI;NOZU KOHEI;HASHIZUME HIROSHI;TADANO GENTA;SATO JUN;TAMURA YUUSUKE;MITSUOKA YASUNORI;ONCOTHERAPY SCIENCE, INC. 发明人 KUSAKABE KEN-ICHI;YOSHIDA HIROSHI;NOZU KOHEI;HASHIZUME HIROSHI;TADANO GENTA;SATO JUN;TAMURA YUUSUKE;MITSUOKA YASUNORI
分类号 C07D487/04;C07D498/04 主分类号 C07D487/04
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