发明名称 Crystalline forms of rosuvastatin calcium salt
摘要 Bis[(E)-7-[4-(4-fluorophenyl)-6-isopropyl-2-[methyl(methylsulfonyl)amino]pyrimidin-5-yl]-(3R,5S)-3,5-dihydroxyhept-6-enoic acid] (also known as rosuvastatin) calcium salt and hydrates can exist in new crystal forms B and C. These crystal forms provide a higher diversity on crystalline materials to optimize manufacture, formulation and biological efficiency.
申请公布号 US7932387(B2) 申请公布日期 2011.04.26
申请号 US20060883008 申请日期 2006.01.23
申请人 BASF SE 发明人 BLATTER FRITZ;VAN DER SCHAAF PAUL ADRIAAN;SZELAGIEWICZ MARTIN
分类号 C07D239/42;A61K31/505;A61P3/06 主分类号 C07D239/42
代理机构 代理人
主权项
地址