发明名称 |
PYRAZOLECARBOXYLIC ACID DERIVATIVES, THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
摘要 |
The invention concerns N-piperidino-5-(4-bromophenyl)-1- (2,4dichlorophenyl)-4-ethylpyrazole-3-carboxamide of formula (I), (See formula I) the salts and solvents thereof which are powerful antagonists of cannabinoid CB 1 receptors. The method for preparing them consists in reacting a functional derivative of 5-(4- brothophenyl)-1-(2,4-dichlorophenyl)-4-ethylpyrazole-3-carboxylic acid with 1-aminopiperidine with subsequent optional salification.
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申请公布号 |
CA2358885(C) |
申请公布日期 |
2007.04.17 |
申请号 |
CA20002358885 |
申请日期 |
2000.01.28 |
申请人 |
SANOFI-SYNTHELABO |
发明人 |
CAMUS, PHILIPPE;MARTINEZ, SERGE;RINALDI, MURIELLE;BARTH, FRANCIS |
分类号 |
C07D231/14;A61K31/415;A61K31/454;A61P3/00;A61P3/04;A61P25/00;A61P25/18;A61P25/28;A61P25/32;A61P25/34;A61P43/00;C07C69/738;C07C251/80 |
主分类号 |
C07D231/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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