发明名称 Compounds as tyrosine kinase modulators
摘要 Disclosed is a compound represented by Formula 1 e.g. [({ 5-[4-(2-fluoro-5-{ [(2-fluoro-5-methylphenyl)amino]carbonyl} phenoxy)pyridin-2-yl]-1H-pyrrol-3-yl} carbonyl)amino]acetic acid wherein for the treatment of one of the diseases or conditions selected from the group consisting of colorectal cancer, lung cancer, hematological cancer, renal cancer, liver cancer, breast cancer, diabetic retinopathy, macular degeneration, age-related macular degeneration, retinopathy of prematurity, ocular angiogenesis, retinal edema, retinal ischemia, diabetic macular edema, cystoid macular edema, retinal vein occlusion, branch vein occlusion, preretinal neovascularization, laser-induced choroidal neovascularization, neovascularization associated with keratoplasty, glaucoma and ocular tumors, arthritis, restenosis, hepatic cirrhosis, atherosclerosis, psoriasis, diabetes mellitus, wound healing, inflammation, neurodegenerative diseases and immune disorders in the human being.
申请公布号 NZ598781(A) 申请公布日期 2014.05.30
申请号 NZ20100598781 申请日期 2010.09.03
申请人 ALLERGAN INC. 发明人 GUO XIALING;ZHU ZHEN
分类号 C07D401/04;A61K31/443;A61K31/4436;A61K31/4439;A61P3/10;A61P27/02;A61P29/00;A61P35/00;C07D401/14;C07D405/14;C07D409/04;C07D409/14 主分类号 C07D401/04
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