发明名称 STABILIZED CRYSTAL OF TIPIRACIL HYDROCHLORIDE, AND CRYSTALLIZATION METHOD FOR SAME
摘要 The present invention addresses the problem of producing a stabilized crystal of 5-chloro-6-[(2- iminopyrrolidin-1-yl)methyl]pyrimidine-2,4(1H,3H)-dione monohydrochloride. As a means for solving the problem, a crystal of 5-chloro-6-[(2-iminopyrrolidin-1-yl)methyl]pyrimidine-2,4(1H,3H)-dione monohydrochloride is provided. The crystal has characteristic peaks at diffraction angles (2&thetas; ± 0.1˚) of 11.6˚, 17.2˚, 17.8˚, 23.3˚, 27.1˚ and 29.3˚ in powder X-ray diffraction.
申请公布号 WO2014203877(A1) 申请公布日期 2014.12.24
申请号 WO2014JP65985 申请日期 2014.06.17
申请人 TAIHO PHARMACEUTICAL CO., LTD. 发明人 KAZUNO, HIDEKI;MUTSUMI, TOMONOBU
分类号 C07D403/06;A61K31/506;A61K31/7072;A61P35/00;A61P43/00 主分类号 C07D403/06
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